In vitro and in vivo characterization of conantokin-R, a selective NMDA receptor antagonist isolated from the venom of the fish-hunting snail Conus radiatus. [electronic resource]
- The Journal of pharmacology and experimental therapeutics Jan 2000
- 425-32 p. digital
Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, P.H.S.
0022-3565
Animals Anticonvulsants--therapeutic use Behavior, Animal--drug effects Binding, Competitive Cerebral Cortex--drug effects Conotoxins--chemical synthesis Dizocilpine Maleate--therapeutic use Dose-Response Relationship, Drug Drug Interactions Electroshock Evoked Potentials--drug effects Female Glutamic Acid--pharmacology In Vitro Techniques Kainic Acid--pharmacology Male Mice Mollusk Venoms--chemistry Oocytes--physiology Pentylenetetrazole--toxicity Piperidines--therapeutic use Receptors, AMPA--classification Receptors, N-Methyl-D-Aspartate--antagonists & inhibitors Recombinant Proteins Seizures--drug therapy Sound--adverse effects Xenopus--physiology gamma-Aminobutyric Acid--pharmacology