Renau, T E

Inhibitors of efflux pumps in Pseudomonas aeruginosa potentiate the activity of the fluoroquinolone antibacterial levofloxacin. [electronic resource] - Journal of medicinal chemistry Dec 1999 - 4928-31 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

0022-2623

10.1021/jm9904598 doi


Anti-Infective Agents--pharmacology
Bacterial Outer Membrane Proteins--antagonists & inhibitors
Carrier Proteins--antagonists & inhibitors
Dipeptides--chemical synthesis
Drug Resistance, Microbial
Drug Stability
Drug Synergism
Endopeptidases--metabolism
Gene Expression
Levofloxacin
Membrane Transport Proteins
Molecular Structure
Ofloxacin--pharmacology
Ornithine--chemistry
Pseudomonas aeruginosa--drug effects
Structure-Activity Relationship