Chin, C N

The third transmembrane helix of the cannabinoid receptor plays a role in the selectivity of aminoalkylindoles for CB2, peripheral cannabinoid receptor. [electronic resource] - The Journal of pharmacology and experimental therapeutics Nov 1999 - 837-44 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, P.H.S.

0022-3565


Animals
Benzoxazines
Binding Sites
CHO Cells--physiology
Central Nervous System--physiology
Cloning, Organism
Colforsin--pharmacology
Cricetinae
Cyclic AMP--metabolism
DNA, Complementary--genetics
Dose-Response Relationship, Drug
Humans
In Vitro Techniques
Indoles--metabolism
Ligands
Morpholines--metabolism
Mutagenesis
Naphthalenes--metabolism
Plasmids
Protein Binding
Receptors, Cannabinoid
Receptors, Drug--chemistry
Recombinant Fusion Proteins--metabolism
Spleen--physiology