The third transmembrane helix of the cannabinoid receptor plays a role in the selectivity of aminoalkylindoles for CB2, peripheral cannabinoid receptor. [electronic resource]
- The Journal of pharmacology and experimental therapeutics Nov 1999
- 837-44 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, P.H.S.
0022-3565
Animals Benzoxazines Binding Sites CHO Cells--physiology Central Nervous System--physiology Cloning, Organism Colforsin--pharmacology Cricetinae Cyclic AMP--metabolism DNA, Complementary--genetics Dose-Response Relationship, Drug Humans In Vitro Techniques Indoles--metabolism Ligands Morpholines--metabolism Mutagenesis Naphthalenes--metabolism Plasmids Protein Binding Receptors, Cannabinoid Receptors, Drug--chemistry Recombinant Fusion Proteins--metabolism Spleen--physiology