Bom, D

Novel A,B,E-ring-modified camptothecins displaying high lipophilicity and markedly improved human blood stabilities. [electronic resource] - Journal of medicinal chemistry Aug 1999 - 3018-22 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, P.H.S.

0022-2623

10.1021/jm9902279 doi


Camptothecin--analogs & derivatives
Chromatography, High Pressure Liquid
Dimyristoylphosphatidylcholine--chemistry
Drug Stability
Enzyme Inhibitors--chemical synthesis
Fluorescence Polarization
Humans
Hydrolysis
Phosphatidylglycerols--chemistry
Spectrometry, Fluorescence
Structure-Activity Relationship
Topoisomerase I Inhibitors