Nassif-Makki, T

Bisquaternary ligands of the common allosteric site of M2 acetylcholine receptors: search for the minimum essential distances between the pharmacophoric elements. [electronic resource] - Journal of medicinal chemistry Mar 1999 - 849-58 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

0022-2623

10.1021/jm981023f doi


Allosteric Site
Animals
Hydrolysis
In Vitro Techniques
Kinetics
Ligands
Models, Molecular
Myocardium--metabolism
Phthalimides--chemical synthesis
Pyridines--chemical synthesis
Radioligand Assay
Receptors, Muscarinic--metabolism
Structure-Activity Relationship
Swine