Li, A H Synthesis, CoMFA analysis, and receptor docking of 3,5-diacyl-2, 4-dialkylpyridine derivatives as selective A3 adenosine receptor antagonists. [electronic resource] - Journal of medicinal chemistry Feb 1999 - 706-21 p. digital Publication Type: Journal Article ISSN: 0022-2623 Standard No.: 10.1021/jm980550w doi Subjects--Topical Terms: AnimalsBinding SitesBinding, CompetitiveBridged Bicyclo Compounds, Heterocyclic--chemical synthesisCHO CellsCell LineCerebral Cortex--metabolismCricetinaeHumansIn Vitro TechniquesLigandsMiceModels, MolecularNeostriatum--metabolismPurinergic P1 Receptor AgonistsRadioligand AssayRatsReceptor, Adenosine A3Receptors, Purinergic P1--metabolismRecombinant Proteins--agonistsStructure-Activity Relationship