5-Fluoro-2-methyl-N-[4-(5H-pyrrolo[2,1-c]-[1, 4]benzodiazepin-10(11H)-ylcarbonyl)-3-chlorophenyl]benzamide (VPA-985): an orally active arginine vasopressin antagonist with selectivity for V2 receptors. [electronic resource]
Producer: 19980724Description: 2442-4 p. digitalISSN:- 0022-2623
- Administration, Oral
- Animals
- Arginine Vasopressin -- antagonists & inhibitors
- Azepines -- administration & dosage
- Benzamides -- administration & dosage
- Blood Platelets -- metabolism
- Body Water -- metabolism
- Cell Line
- Cell Membrane -- metabolism
- Dogs
- Fibroblasts -- drug effects
- Humans
- Kidney -- metabolism
- Liver -- metabolism
- Osmolar Concentration
- Pyrroles
- Rats
- Receptors, Vasopressin -- metabolism
- Sodium -- blood
- Structure-Activity Relationship
- Urine -- chemistry
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Publication Type: Clinical Trial; Journal Article; Randomized Controlled Trial
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