Development of orally active oxytocin antagonists: studies on 1-(1-[4-[1-(2-methyl-1-oxidopyridin-3-ylmethyl)piperidin-4-yloxy]-2- methoxybenzoyl]piperidin-4-yl)-1,4-dihydrobenz[d][1,3]oxazin-2-one (L-372,662) and related pyridines. [electronic resource]
Producer: 19980624Description: 2146-63 p. digitalISSN:- 0022-2623
- Administration, Oral
- Animals
- Biological Availability
- Cell Line
- Chromatography, High Pressure Liquid
- Dogs
- Female
- Humans
- Kidney -- cytology
- Liver -- metabolism
- Male
- Mass Spectrometry
- Oxazines -- chemical synthesis
- Pregnancy
- Pyridines -- chemical synthesis
- Rats
- Receptors, Oxytocin -- antagonists & inhibitors
- Recombinant Proteins -- antagonists & inhibitors
- Spectrophotometry, Ultraviolet
- Uterine Contraction -- drug effects
- Uterus -- drug effects
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Publication Type: Comparative Study; Journal Article
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