Deramciclane, a putative anxiolytic drug, is a serotonin 5-HT2C receptor inverse agonist but fails to induce 5-HT2C receptor down-regulation. [electronic resource]
Producer: 19980618Description: 99-104 p. digitalISSN:- 0033-3158
- Animals
- Anti-Anxiety Agents -- pharmacology
- Brain -- drug effects
- Camphanes -- pharmacology
- Clozapine -- pharmacology
- Inositol Phosphates -- metabolism
- Male
- Rats
- Rats, Sprague-Dawley
- Receptor, Serotonin, 5-HT2A
- Receptor, Serotonin, 5-HT2C
- Receptors, Serotonin -- drug effects
- Serotonin Antagonists -- pharmacology
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Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't
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