4-Amino-2-[4-[1-(benzyloxycarbonyl)-2(S)- [[(1,1-dimethylethyl)amino]carbonyl]-piperazinyl]-6, 7-dimethoxyquinazoline (L-765,314): a potent and selective alpha1b adrenergic receptor antagonist. [electronic resource]
Producer: 19980501Description: 1205-8 p. digitalISSN:- 0022-2623
- Adrenergic alpha-1 Receptor Antagonists
- Adrenergic alpha-Antagonists -- chemical synthesis
- Animals
- Antihypertensive Agents -- chemical synthesis
- Blood Pressure -- drug effects
- Humans
- Male
- Organ Specificity
- Prazosin -- analogs & derivatives
- Rats
- Rats, Inbred SHR
- Rats, Sprague-Dawley
- Receptors, Adrenergic, alpha-1 -- metabolism
- Spinal Cord -- metabolism
- Structure-Activity Relationship
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Publication Type: Comparative Study; Journal Article
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