Targeting delavirdine/atevirdine resistant HIV-1: identification of (alkylamino)piperidine-containing bis(heteroaryl)piperazines as broad spectrum HIV-1 reverse transcriptase inhibitors. [electronic resource]
Producer: 19961104Description: 3769-89 p. digitalISSN:- 0022-2623
- Animals
- Anti-HIV Agents -- chemical synthesis
- Biological Availability
- Cell Line
- Delavirdine
- Drug Resistance, Microbial
- Drug Stability
- HIV Reverse Transcriptase
- HIV-1 -- drug effects
- Indoles -- pharmacology
- Molecular Structure
- Piperazines -- pharmacology
- Piperidines -- chemical synthesis
- Pyridines -- chemical synthesis
- Rats
- Reverse Transcriptase Inhibitors -- chemical synthesis
- Structure-Activity Relationship
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Publication Type: Comparative Study; Journal Article
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