Characterization of irreversible binding of beta-funaltrexamine to the cloned rat mu opioid receptor. [electronic resource]
Producer: 19950905Description: 17866-70 p. digitalISSN:- 0021-9258
- 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer
- Amino Acid Sequence
- Animals
- Cell Line
- Cloning, Molecular
- Diprenorphine -- metabolism
- Electrophoresis, Polyacrylamide Gel
- Enkephalin, Leucine -- analogs & derivatives
- Glycosylation
- Molecular Sequence Data
- Naltrexone -- analogs & derivatives
- Oligopeptides -- pharmacology
- Protein Binding
- Pyrrolidines -- pharmacology
- Rats
- Rats, Sprague-Dawley
- Receptors, Opioid, delta -- drug effects
- Receptors, Opioid, kappa -- antagonists & inhibitors
- Receptors, Opioid, mu -- antagonists & inhibitors
- Recombinant Proteins -- metabolism
- Sodium -- metabolism
- Tritium
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Publication Type: Journal Article; Research Support, U.S. Gov't, P.H.S.
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