In vitro and in vivo evidence for a tachykinin NK1 receptor antagonist effect of vapreotide, an analgesic cyclic analog of somatostatin. [electronic resource]
Producer: 19951106Description: 241-9 p. digitalISSN:- 0014-2999
- Acetylcholine -- pharmacology
- Analgesics -- metabolism
- Animals
- Binding, Competitive -- drug effects
- Brain -- metabolism
- Bronchi -- drug effects
- Capillary Permeability -- drug effects
- Duodenum -- drug effects
- Electric Stimulation
- Female
- Guinea Pigs
- In Vitro Techniques
- Injections, Spinal
- Male
- Mice
- Muscle Contraction -- drug effects
- Muscle, Smooth -- drug effects
- Neurokinin A -- analogs & derivatives
- Neurokinin-1 Receptor Antagonists
- Peptide Fragments -- pharmacology
- Rats
- Rats, Sprague-Dawley
- Receptors, Neurokinin-1 -- metabolism
- Somatostatin -- analogs & derivatives
- Substance P -- metabolism
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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