Allosteric p97 Inhibitors Can Overcome Resistance to ATP-Competitive p97 Inhibitors for Potential Anticancer Therapy. [electronic resource]
Producer: 20210520Description: 685-694 p. digitalISSN:- 1860-7187
- Acetanilides -- chemistry
- Adenosine Triphosphatases -- antagonists & inhibitors
- Adenosine Triphosphate -- metabolism
- Allosteric Regulation -- drug effects
- Antineoplastic Agents -- chemistry
- Benzothiazoles -- chemistry
- Cell Proliferation -- drug effects
- Dose-Response Relationship, Drug
- Drug Resistance, Neoplasm -- drug effects
- Drug Screening Assays, Antitumor
- Enzyme Inhibitors -- chemistry
- HCT116 Cells
- Humans
- Indoles -- chemistry
- Models, Molecular
- Molecular Structure
- Nuclear Proteins -- antagonists & inhibitors
- Pyrimidines -- chemistry
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Publication Type: Journal Article; Research Support, N.I.H., Extramural
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