Allosteric modulators restore orthosteric agonist binding to mutated CB [electronic resource]
Producer: 20200601Description: 84-91 p. digitalISSN:- 2042-7158
- Binding Sites
- Cannabinoid Receptor Agonists -- metabolism
- Cyclohexanols -- metabolism
- HEK293 Cells
- Humans
- Indoles -- metabolism
- Ligands
- Mutation
- Phenylurea Compounds -- metabolism
- Piperidines -- metabolism
- Protein Binding
- Protein Conformation
- Pyridines -- metabolism
- Receptor, Cannabinoid, CB1 -- agonists
- Rimonabant -- metabolism
- Structure-Activity Relationship
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Publication Type: Journal Article
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