Improved Prediction of in Vivo Supersaturation and Precipitation of Poorly Soluble Weakly Basic Drugs Using a Biorelevant Bicarbonate Buffer in a Gastrointestinal Transfer Model. [electronic resource]
Producer: 20200608Description: 3938-3947 p. digitalISSN:- 1543-8392
- Administration, Oral
- Animals
- Bicarbonates -- chemistry
- Buffers
- Chemical Precipitation -- drug effects
- Drug Delivery Systems -- methods
- Drug Liberation -- physiology
- Female
- Gastrointestinal Absorption -- physiology
- Gastrointestinal Tract
- Hydrogen-Ion Concentration
- Indazoles
- Ketoconazole -- administration & dosage
- Lapatinib -- administration & dosage
- Methylcellulose -- analogs & derivatives
- Models, Biological
- Phosphates -- chemistry
- Pyrimidines -- administration & dosage
- Rats
- Rats, Wistar
- Solubility
- Sulfonamides -- administration & dosage
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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