Multiple administrations of fluconazole increase plasma exposure to ruxolitinib in healthy adult subjects. [electronic resource]
Producer: 20200512Description: 749-757 p. digitalISSN:- 1432-0843
- Adult
- Cytochrome P-450 CYP2C9 -- metabolism
- Cytochrome P-450 CYP3A -- metabolism
- Dose-Response Relationship, Drug
- Drug Administration Schedule
- Drug Interactions
- Enzyme Inhibitors -- pharmacokinetics
- Female
- Fluconazole -- pharmacokinetics
- Half-Life
- Healthy Volunteers
- Humans
- Janus Kinases -- metabolism
- Male
- Metabolic Clearance Rate -- drug effects
- Middle Aged
- Nitriles
- Pyrazoles -- pharmacokinetics
- Pyrimidines
- Signal Transduction -- drug effects
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Publication Type: Clinical Trial, Phase I; Journal Article; Research Support, Non-U.S. Gov't
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