First-in-human phase 1 study of novel dUTPase inhibitor TAS-114 in combination with S-1 in Japanese patients with advanced solid tumors. [electronic resource]
Producer: 20200220Description: 507-518 p. digitalISSN:- 1573-0646
- Adult
- Aged
- Aged, 80 and over
- Antimetabolites, Antineoplastic -- pharmacokinetics
- Drug Combinations
- Drug Therapy, Combination
- Enzyme Inhibitors -- pharmacokinetics
- Female
- Follow-Up Studies
- Humans
- Male
- Maximum Tolerated Dose
- Middle Aged
- Neoplasms -- drug therapy
- Oxonic Acid -- pharmacokinetics
- Prognosis
- Pyrimidines -- pharmacokinetics
- Pyrophosphatases -- antagonists & inhibitors
- Sulfonamides -- pharmacokinetics
- Tegafur -- pharmacokinetics
- Tissue Distribution
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Publication Type: Clinical Trial, Phase I; Journal Article; Multicenter Study; Research Support, Non-U.S. Gov't
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