2-Acyl-3-carboxyl-tetrahydroisoquinoline Derivatives: Mixed-Type PTP1B Inhibitors without PPARγ Activation. [electronic resource]
Producer: 20181224Description: 1131-1152 p. digitalISSN:- 1347-5223
- Animals
- Diabetes Mellitus, Experimental -- drug therapy
- Dose-Response Relationship, Drug
- Enzyme Inhibitors -- blood
- Humans
- Hypoglycemic Agents -- blood
- Male
- Mice
- Mice, Inbred Strains
- Molecular Docking Simulation
- Molecular Structure
- PPAR gamma -- metabolism
- Protein Tyrosine Phosphatase, Non-Receptor Type 1 -- antagonists & inhibitors
- Rats
- Rats, Sprague-Dawley
- Structure-Activity Relationship
- Tetrahydroisoquinolines -- blood
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Publication Type: Journal Article
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