Characterization and inhibition of mephenytoin 4-hydroxylase activity in human liver microsomes. [electronic resource]
Producer: 19870227Description: 216-22 p. digitalISSN:- 0022-3565
- Anticonvulsants -- metabolism
- Aryl Hydrocarbon Hydroxylases
- Binding, Competitive
- Cytochrome P-450 CYP2C19
- Cytochrome P-450 Enzyme System -- metabolism
- Humans
- Hydantoins -- metabolism
- Isoenzymes -- metabolism
- Kinetics
- Mephenytoin -- metabolism
- Microsomes, Liver -- enzymology
- Mixed Function Oxygenases -- antagonists & inhibitors
- NADP -- metabolism
- Phenytoin -- metabolism
- Polymorphism, Genetic
- Stereoisomerism
- Warfarin -- pharmacology
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Publication Type: Journal Article; Research Support, U.S. Gov't, P.H.S.
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