In Silico Design and Enantioselective Synthesis of Functionalized Monocyclic 3-Amino-1-carboxymethyl-β-lactams as Inhibitors of Penicillin-Binding Proteins of Resistant Bacteria. [electronic resource]
Producer: 20181024Description: 15254-15266 p. digitalISSN:- 1521-3765
- Amination
- Anti-Bacterial Agents -- chemical synthesis
- Bacterial Infections -- drug therapy
- Computer Simulation
- Computer-Aided Design
- Drug Design
- Drug Resistance, Bacterial -- drug effects
- Enterococcus faecium -- drug effects
- Escherichia coli -- drug effects
- Escherichia coli Infections -- drug therapy
- Gram-Positive Bacterial Infections -- drug therapy
- Humans
- Molecular Docking Simulation
- Penicillin-Binding Proteins -- antagonists & inhibitors
- beta-Lactams -- chemical synthesis
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Publication Type: Journal Article
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