Virtual Fragment Screening Identification of a Quinoline-5,8-dicarboxylic Acid Derivative as a Selective JMJD3 Inhibitor. [electronic resource]
Producer: 20190715Description: 1160-1164 p. digitalISSN:- 1860-7187
- Binding Sites
- Dicarboxylic Acids -- chemical synthesis
- Enzyme Inhibitors -- chemical synthesis
- Humans
- Isoenzymes -- antagonists & inhibitors
- Jumonji Domain-Containing Histone Demethylases -- antagonists & inhibitors
- Molecular Docking Simulation
- Molecular Dynamics Simulation
- Quinolines -- chemical synthesis
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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