Discovery of 7-Oxo-2,4,5,7-tetrahydro-6 H-pyrazolo[3,4- c]pyridine Derivatives as Potent, Orally Available, and Brain-Penetrating Receptor Interacting Protein 1 (RIP1) Kinase Inhibitors: Analysis of Structure-Kinetic Relationships. [electronic resource]
Producer: 20190417Description: 2384-2409 p. digitalISSN:- 1520-4804
- Animals
- Brain -- metabolism
- Cell Death -- drug effects
- Cell Line
- Encephalomyelitis, Autoimmune, Experimental -- drug therapy
- High-Throughput Screening Assays
- Humans
- Mice
- Models, Molecular
- Molecular Docking Simulation
- Necrosis
- Nuclear Pore Complex Proteins -- antagonists & inhibitors
- Protein Kinase Inhibitors -- chemical synthesis
- Pyridines -- chemical synthesis
- RNA-Binding Proteins -- antagonists & inhibitors
- Structure-Activity Relationship
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Publication Type: Journal Article
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