Intestinal absorption and activation of decitabine amino acid ester prodrugs mediated by peptide transporter PEPT1 and enterocyte enzymes. [electronic resource]
Producer: 20180907Description: 64-71 p. digitalISSN:- 1873-3476
- Administration, Oral
- Amino Acids -- chemistry
- Animals
- Azacitidine -- administration & dosage
- Biological Availability
- Cell Membrane Permeability
- DNA Modification Methylases -- antagonists & inhibitors
- Decitabine
- Enterocytes -- enzymology
- Enzyme Inhibitors -- pharmacokinetics
- Esters -- chemistry
- Intestinal Absorption
- Intestinal Mucosa -- metabolism
- Intestines -- cytology
- Male
- Models, Animal
- Peptide Transporter 1 -- metabolism
- Prodrugs -- administration & dosage
- Rats
- Rats, Sprague-Dawley
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Publication Type: Journal Article
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