Host-parasite co-metabolic activation of antitrypanosomal aminomethyl-benzoxaboroles. [electronic resource]
Producer: 20180622Description: e1006850 p. digitalISSN:- 1553-7374
- Activation, Metabolic
- Aldehyde Dehydrogenase -- antagonists & inhibitors
- Aldehyde Oxidoreductases -- antagonists & inhibitors
- Amine Oxidase (Copper-Containing) -- antagonists & inhibitors
- Amino Acid Substitution
- Animals
- Boron Compounds -- chemistry
- Drug Resistance
- High-Throughput Screening Assays
- Humans
- Models, Biological
- Molecular Structure
- Mutation
- Phylogeny
- Prodrugs -- chemistry
- Protein Interaction Domains and Motifs
- RNA Interference
- Rats
- Recombinant Fusion Proteins -- chemistry
- Recombinant Proteins -- chemistry
- Structure-Activity Relationship
- Trypanocidal Agents -- chemistry
- Trypanosoma brucei brucei -- drug effects
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Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't
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