Fragment-based discovery of a potent NAMPT inhibitor. [electronic resource]
Producer: 20190530Description: 437-440 p. digitalISSN:- 1464-3405
- Acrylamides -- chemical synthesis
- Cytokines -- antagonists & inhibitors
- Dose-Response Relationship, Drug
- Drug Discovery
- Drug Evaluation, Preclinical
- Enzyme Inhibitors -- chemical synthesis
- Fluorescence Resonance Energy Transfer
- Humans
- Molecular Docking Simulation
- Molecular Structure
- Nicotinamide Phosphoribosyltransferase -- antagonists & inhibitors
- Piperidines -- chemical synthesis
- Structure-Activity Relationship
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Publication Type: Journal Article; Research Support, U.S. Gov't, Non-P.H.S.
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