Characterization of isoflavonoids as inhibitors of β-hydroxyacyl-acyl carrier protein dehydratase (FabZ) from Moraxella catarrhalis: Kinetics, spectroscopic, thermodynamics and in silico studies. [electronic resource]
Producer: 20180522Description: 726-744 p. digitalISSN:- 0304-4165
- Acyl Coenzyme A -- metabolism
- Amino Acid Sequence
- Bacterial Proteins -- antagonists & inhibitors
- Binding Sites -- drug effects
- Catalytic Domain -- drug effects
- Circular Dichroism
- Conserved Sequence
- Drug Design
- Drug Resistance, Multiple, Bacterial
- Flavonoids -- pharmacology
- Genistein -- pharmacology
- Hydro-Lyases -- antagonists & inhibitors
- Hydrogen-Ion Concentration
- Isoflavones -- pharmacology
- Kinetics
- Microbial Sensitivity Tests
- Models, Molecular
- Molecular Dynamics Simulation
- Molecular Structure
- Moraxella catarrhalis -- drug effects
- Phylogeny
- Protein Conformation
- Recombinant Proteins -- chemistry
- Sequence Alignment
- Spectrometry, Fluorescence
- Structure-Activity Relationship
- Temperature
- Thermodynamics
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Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't
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