Structure-Activity Relationship Studies of β-Lactam-azide Analogues as Orally Active Antitumor Agents Targeting the Tubulin Colchicine Site. [electronic resource]
Producer: 20190625Description: 12788 p. digitalISSN:- 2045-2322
- Administration, Oral
- Animals
- Antineoplastic Agents -- administration & dosage
- Apoptosis -- drug effects
- Azides -- administration & dosage
- Cadherins -- metabolism
- Cell Line, Tumor
- Cell Movement -- drug effects
- Colchicine -- chemistry
- Down-Regulation -- drug effects
- Humans
- Inhibitory Concentration 50
- Mice, Inbred BALB C
- Mice, Nude
- Structure-Activity Relationship
- Tubulin -- metabolism
- Up-Regulation -- drug effects
- Zonula Occludens-1 Protein -- metabolism
- beta-Lactams -- administration & dosage
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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