Novel Chemical Scaffolds for Inhibition of Rifamycin-Resistant RNA Polymerase Discovered from High-Throughput Screening. [electronic resource]
Producer: 20181231Description: 287-297 p. digitalISSN:- 2472-5560
- Antitubercular Agents -- pharmacology
- Aptamers, Nucleotide -- genetics
- Bacterial Proteins -- antagonists & inhibitors
- Biological Assay
- DNA-Directed RNA Polymerases -- antagonists & inhibitors
- Drug Discovery
- Drug Resistance, Bacterial -- drug effects
- Escherichia coli -- drug effects
- Extensively Drug-Resistant Tuberculosis -- drug therapy
- Gene Expression
- High-Throughput Screening Assays
- Humans
- Microbial Sensitivity Tests
- Mutation
- Mycobacterium tuberculosis -- drug effects
- Plasmids -- chemistry
- Rifampin -- pharmacology
- Rifamycins -- pharmacology
- Small Molecule Libraries -- chemistry
- Structure-Activity Relationship
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Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
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