The consequence of regional gradients of P-gp and CYP3A4 for drug-drug interactions by P-gp inhibitors and the P-gp/CYP3A4 interplay in the human intestine ex vivo. [electronic resource]
Producer: 20170726Description: 26-33 p. digitalISSN:- 1879-3177
- ATP Binding Cassette Transporter, Subfamily B, Member 1 -- antagonists & inhibitors
- Adult
- Aged
- Aged, 80 and over
- Colon -- metabolism
- Cyclosporins -- pharmacology
- Cytochrome P-450 CYP3A -- metabolism
- Cytochrome P-450 CYP3A Inhibitors -- pharmacology
- Drug Interactions
- Female
- Humans
- Ileum -- metabolism
- In Vitro Techniques
- Isoquinolines -- pharmacology
- Jejunum -- metabolism
- Ketoconazole -- pharmacology
- Male
- Middle Aged
- Quinazolines -- pharmacology
- Quinidine -- analogs & derivatives
- Verapamil -- pharmacology
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Publication Type: Journal Article
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