Tamoxifen Isomers and Metabolites Exhibit Distinct Affinity and Activity at Cannabinoid Receptors: Potential Scaffold for Drug Development. [electronic resource]
Producer: 20170726Description: e0167240 p. digitalISSN:- 1932-6203
- Adenylyl Cyclases -- metabolism
- Animals
- Binding, Competitive
- Breast Neoplasms -- drug therapy
- CHO Cells
- Cannabinoid Receptor Agonists -- metabolism
- Cannabinoid Receptor Antagonists -- metabolism
- Colforsin -- metabolism
- Cricetinae
- Cricetulus
- Cyclic AMP -- metabolism
- Cyclohexanols -- metabolism
- Female
- GTP-Binding Proteins -- metabolism
- Guanosine 5'-O-(3-Thiotriphosphate) -- metabolism
- Humans
- Indoles -- metabolism
- Isomerism
- Receptor, Cannabinoid, CB1 -- agonists
- Receptor, Cannabinoid, CB2 -- agonists
- Selective Estrogen Receptor Modulators -- chemistry
- Tamoxifen -- analogs & derivatives
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Publication Type: Journal Article
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