The Bruton Tyrosine Kinase (BTK) Inhibitor Acalabrutinib Demonstrates Potent On-Target Effects and Efficacy in Two Mouse Models of Chronic Lymphocytic Leukemia. [electronic resource]
Producer: 20180316Description: 2831-2841 p. digitalISSN:- 1557-3265
- Adenine -- analogs & derivatives
- Adoptive Transfer -- methods
- Agammaglobulinaemia Tyrosine Kinase
- Animals
- Antineoplastic Combined Chemotherapy Protocols -- administration & dosage
- Apoptosis -- drug effects
- Benzamides -- administration & dosage
- Disease Models, Animal
- Humans
- Leukemia, Lymphocytic, Chronic, B-Cell -- drug therapy
- Mice
- Mice, Transgenic
- Piperidines
- Protein Kinase Inhibitors -- administration & dosage
- Protein-Tyrosine Kinases -- antagonists & inhibitors
- Proto-Oncogene Proteins -- genetics
- Pyrazines -- administration & dosage
- Pyrazoles -- administration & dosage
- Pyrimidines -- administration & dosage
- Xenograft Model Antitumor Assays
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Publication Type: Journal Article
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