Discovery of Imidazoquinolines as a Novel Class of Potent, Selective, and in Vivo Efficacious Cancer Osaka Thyroid (COT) Kinase Inhibitors. [electronic resource]
Producer: 20170606Description: 7544-60 p. digitalISSN:- 1520-4804
- Animals
- Crystallography, X-Ray
- Dogs
- Dose-Response Relationship, Drug
- Drug Discovery
- Humans
- Imidazoles -- chemical synthesis
- MAP Kinase Kinase Kinases -- antagonists & inhibitors
- Male
- Models, Molecular
- Molecular Structure
- Protein Kinase Inhibitors -- chemical synthesis
- Proto-Oncogene Proteins -- antagonists & inhibitors
- Quinolines -- chemical synthesis
- Rats
- Rats, Sprague-Dawley
- Structure-Activity Relationship
- Tumor Necrosis Factor-alpha -- antagonists & inhibitors
No physical items for this record
Publication Type: Journal Article
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