Synthesis and in vivo Evaluation of Fluorine-18 and Iodine-123 Pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine Derivatives as PET and SPECT Radiotracers for Mapping A2A Receptors. [electronic resource]
Producer: 20170519Description: 1936-43 p. digitalISSN:- 1860-7187
- Animals
- Brain -- diagnostic imaging
- Dose-Response Relationship, Drug
- Female
- Fluorine Radioisotopes
- Heterocyclic Compounds, 3-Ring -- chemical synthesis
- Humans
- Iodine Isotopes
- Macaca mulatta
- Molecular Conformation
- Papio
- Positron-Emission Tomography
- Pyrimidines -- chemical synthesis
- Radioactive Tracers
- Radiopharmaceuticals -- chemical synthesis
- Receptor, Adenosine A2A -- chemistry
- Recombinant Proteins -- chemistry
- Structure-Activity Relationship
- Triazoles -- chemical synthesis
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Publication Type: Journal Article
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