Role of the Substrate Specificity-Defining Residues of Human SIRT5 in Modulating the Structural Stability and Inhibitory Features of the Enzyme. [electronic resource]
Producer: 20160829Description: e0152467 p. digitalISSN:- 1932-6203
- Amino Acids -- metabolism
- Biocatalysis -- drug effects
- Calorimetry
- Carbazoles -- chemistry
- Catalytic Domain
- Circular Dichroism
- Enzyme Stability -- drug effects
- Humans
- Kinetics
- Models, Molecular
- Mutant Proteins -- chemistry
- Mutation -- genetics
- Niacinamide -- pharmacology
- Protein Denaturation -- drug effects
- Protein Structure, Secondary
- Sirtuin 1 -- genetics
- Sirtuins -- antagonists & inhibitors
- Structure-Activity Relationship
- Substrate Specificity -- drug effects
- Temperature
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Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, U.S. Gov't, Non-P.H.S.
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