Novel β-Carboline/Hydroxamic Acid Hybrids Targeting Both Histone Deacetylase and DNA Display High Anticancer Activity via Regulation of the p53 Signaling Pathway. [electronic resource]
Producer: 20160412Description: 9214-27 p. digitalISSN:- 1520-4804
- Acetylation -- drug effects
- Animals
- Antineoplastic Agents -- chemistry
- Apoptosis -- drug effects
- Carbolines -- chemistry
- Cell Proliferation -- drug effects
- Colon -- drug effects
- Colorectal Neoplasms -- drug therapy
- DNA -- metabolism
- Female
- HCT116 Cells
- Histone Deacetylase Inhibitors -- chemistry
- Histone Deacetylases -- metabolism
- Humans
- Hydroxamic Acids -- chemistry
- Mice
- Mice, Inbred BALB C
- Mice, Nude
- Rectum -- drug effects
- Signal Transduction -- drug effects
- Tubulin -- metabolism
- Tumor Suppressor Protein p53 -- metabolism
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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