A Nampt inhibitor FK866 mimics vitamin B3 deficiency by causing senescence of human fibroblastic Hs68 cells via attenuation of NAD(+)-SIRT1 signaling. [electronic resource]
Producer: 20160801Description: 789-800 p. digitalISSN:- 1573-6768
- AMP-Activated Protein Kinases -- metabolism
- Acrylamides -- pharmacology
- Cell Line
- Cell Proliferation -- drug effects
- Cellular Senescence -- drug effects
- Cytokines -- antagonists & inhibitors
- Enzyme Inhibitors -- pharmacology
- Fibroblasts -- cytology
- Glutathione -- metabolism
- Humans
- NAD -- metabolism
- NADP -- metabolism
- Niacin -- pharmacology
- Niacinamide -- deficiency
- Nicotinamide Phosphoribosyltransferase -- antagonists & inhibitors
- Piperidines -- pharmacology
- Signal Transduction -- drug effects
- Sirtuin 1 -- metabolism
- TOR Serine-Threonine Kinases -- metabolism
- Tumor Suppressor Protein p53 -- metabolism
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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