CBP30, a selective CBP/p300 bromodomain inhibitor, suppresses human Th17 responses. [electronic resource]
Producer: 20151230Description: 10768-73 p. digitalISSN:- 1091-6490
- Adult
- Aged
- Arthritis, Psoriatic -- metabolism
- Azepines -- pharmacology
- Benzimidazoles -- chemistry
- CD4-Positive T-Lymphocytes -- drug effects
- Calorimetry
- Cells, Cultured
- Crystallography, X-Ray
- Drug Evaluation, Preclinical
- Female
- Gene Expression Regulation -- drug effects
- Humans
- Immunosuppressive Agents -- chemistry
- Interleukin-17 -- biosynthesis
- Isoxazoles -- chemistry
- Kinetics
- Male
- Middle Aged
- Models, Molecular
- Molecular Structure
- Protein Conformation
- Protein Structure, Tertiary -- drug effects
- Recombinant Proteins -- metabolism
- Spondylitis, Ankylosing -- metabolism
- Structure-Activity Relationship
- Th17 Cells -- drug effects
- Triazoles -- pharmacology
- p300-CBP Transcription Factors -- antagonists & inhibitors
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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