Synthesis, Biological, and Computational Evaluation of Novel 1,3,5-Substituted Indolin-2-one Derivatives as Inhibitors of Src Tyrosine Kinase. [electronic resource]
Producer: 20161006Description: 715-29 p. digitalISSN:- 1521-4184
- Drug Design
- Hydrogen Bonding
- Imatinib Mesylate -- pharmacology
- Indoles -- chemical synthesis
- Molecular Docking Simulation
- Molecular Targeted Therapy
- Phosphorylation
- Phosphotyrosine -- metabolism
- Protein Conformation
- Protein Kinase Inhibitors -- chemical synthesis
- Structure-Activity Relationship
- src-Family Kinases -- antagonists & inhibitors
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Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't
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