Novel Octahydropyrrolo[3,4-c]pyrroles Are Selective Orexin-2 Antagonists: SAR Leading to a Clinical Candidate. [electronic resource]
Producer: 20151012Description: 5620-36 p. digitalISSN:- 1520-4804
- Animals
- Clinical Trials as Topic
- Dogs
- Humans
- Intracellular Signaling Peptides and Proteins -- antagonists & inhibitors
- Male
- Neuropeptides -- antagonists & inhibitors
- Orexin Receptors -- metabolism
- Orexins
- Pyrroles -- chemistry
- Rats
- Sleep Initiation and Maintenance Disorders -- drug therapy
- Structure-Activity Relationship
- Substrate Specificity
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Publication Type: Journal Article
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