In vitro cytotoxicity and in vivo efficacy, pharmacokinetics, and metabolism of pyrazole-based small molecule inhibitors of Mdm2/4-p53 interaction. [electronic resource]
Producer: 20151013Description: 287-99 p. digitalISSN:- 1432-0843
- Animals
- Antineoplastic Agents -- chemistry
- Drug Screening Assays, Antitumor
- Female
- HCT116 Cells
- Heterografts
- Humans
- Mice, SCID
- Neoplasm Transplantation
- Proto-Oncogene Proteins -- metabolism
- Proto-Oncogene Proteins c-mdm2 -- metabolism
- Pyrazoles -- chemistry
- Tumor Suppressor Protein p53 -- metabolism
- Ubiquitin-Protein Ligases -- metabolism
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Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
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