Novel inhibitors of cholesterol degradation in Mycobacterium tuberculosis reveal how the bacterium's metabolism is constrained by the intracellular environment. [electronic resource]
Producer: 20160129Description: e1004679 p. digitalISSN:- 1553-7374
- Adenylyl Cyclases -- genetics
- Animals
- Antitubercular Agents -- pharmacology
- Bacterial Proteins -- metabolism
- Cell Line
- Cholesterol -- metabolism
- Cyclic AMP -- metabolism
- Hydroxysteroid Dehydrogenases -- antagonists & inhibitors
- Intracellular Space
- Lipid Metabolism -- drug effects
- Macrophages -- immunology
- Mice
- Microbial Sensitivity Tests
- Mixed Function Oxygenases -- antagonists & inhibitors
- Mycobacterium tuberculosis -- growth & development
- Oxo-Acid-Lyases -- antagonists & inhibitors
- Small Molecule Libraries -- pharmacology
- Tuberculosis, Pulmonary -- drug therapy
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Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
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