A highly potent and selective Vps34 inhibitor alters vesicle trafficking and autophagy. [electronic resource]
Producer: 20150122Description: 1013-9 p. digitalISSN:- 1552-4469
- Adenosine Triphosphate -- chemistry
- Antineoplastic Agents -- chemical synthesis
- Autophagy -- drug effects
- Catalytic Domain
- Cell Line, Tumor
- Cell Proliferation -- drug effects
- Class III Phosphatidylinositol 3-Kinases -- antagonists & inhibitors
- Drug Synergism
- Endosomes -- drug effects
- Everolimus
- Gene Expression
- Humans
- Kidney -- enzymology
- Kinetics
- Lysosomes -- drug effects
- Molecular Docking Simulation
- Protein Kinase Inhibitors -- chemical synthesis
- Pyridines -- chemical synthesis
- Pyrimidinones -- chemical synthesis
- Recombinant Proteins -- chemistry
- Signal Transduction
- Sirolimus -- analogs & derivatives
- TOR Serine-Threonine Kinases -- antagonists & inhibitors
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Publication Type: Journal Article
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