Lapatinib antagonizes multidrug resistance-associated protein 1-mediated multidrug resistance by inhibiting its transport function. [electronic resource]
Producer: 20151208Description: 390-9 p. digitalISSN:- 1528-3658
- Animals
- Antineoplastic Agents -- pharmacology
- Biological Transport -- drug effects
- Cell Line, Tumor
- Cell Survival -- drug effects
- Cisplatin -- pharmacology
- Doxorubicin -- pharmacology
- Drug Resistance, Multiple -- drug effects
- Drug Resistance, Neoplasm -- drug effects
- Drug Synergism
- Extracellular Signal-Regulated MAP Kinases -- metabolism
- HEK293 Cells
- Humans
- Lapatinib
- Mice
- Mice, Nude
- Multidrug Resistance-Associated Protein 2
- Multidrug Resistance-Associated Proteins -- antagonists & inhibitors
- NIH 3T3 Cells
- Neoplasms -- drug therapy
- Proto-Oncogene Proteins c-akt -- metabolism
- Quinazolines -- pharmacology
- Tumor Burden -- drug effects
- Vincristine -- pharmacology
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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