Preclinical characterization of a novel radiolabeled analog of practolol for the molecular imaging of myocardial β-adrenoceptor density. [electronic resource]
Producer: 20150526Description: 984-92 p. digitalISSN:- 1532-6551
- Adrenergic beta-1 Receptor Antagonists -- chemistry
- Animals
- Animals, Newborn
- Cells, Cultured
- Drug Evaluation, Preclinical
- Heart -- diagnostic imaging
- Iodine Radioisotopes -- chemistry
- Isotope Labeling -- methods
- Metabolic Clearance Rate
- Mice
- Molecular Imaging -- methods
- Myocardium -- metabolism
- Myocytes, Cardiac -- diagnostic imaging
- Organ Specificity
- Practolol -- analogs & derivatives
- Radionuclide Imaging
- Radiopharmaceuticals -- chemical synthesis
- Rats
- Receptors, Adrenergic, beta -- metabolism
- Reproducibility of Results
- Sensitivity and Specificity
- Tissue Distribution
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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