Inhibiting Tankyrases sensitizes KRAS-mutant cancer cells to MEK inhibitors via FGFR2 feedback signaling. [electronic resource]
Producer: 20140808Description: 3294-305 p. digitalISSN:- 1538-7445
- Acetamides -- administration & dosage
- Aminopyridines -- administration & dosage
- Aniline Compounds -- administration & dosage
- Animals
- Antineoplastic Combined Chemotherapy Protocols -- pharmacology
- Cell Line, Tumor
- Drug Synergism
- Erlotinib Hydrochloride
- Feedback, Physiological
- Female
- Humans
- MAP Kinase Kinase Kinases -- antagonists & inhibitors
- Mice
- Mice, Nude
- Morpholines -- administration & dosage
- Mutation
- Protein Kinase Inhibitors -- pharmacology
- Proto-Oncogene Proteins -- genetics
- Proto-Oncogene Proteins p21(ras)
- Pyrimidinones -- administration & dosage
- Quinazolines -- administration & dosage
- Receptor, Fibroblast Growth Factor, Type 2 -- antagonists & inhibitors
- Signal Transduction
- Sulfonamides -- administration & dosage
- Tankyrases -- antagonists & inhibitors
- Thiazoles -- administration & dosage
- Xenograft Model Antitumor Assays
- ras Proteins -- genetics
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Publication Type: Journal Article
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