Dolastatin 10, a powerful cytostatic peptide derived from a marine animal. Inhibition of tubulin polymerization mediated through the vinca alkaloid binding domain. [electronic resource]
Producer: 19900719Description: 1941-9 p. digitalISSN:- 0006-2952
- Amino Acid Sequence
- Animals
- Antibiotics, Antineoplastic -- pharmacology
- Aziridines -- pharmacokinetics
- Cell Division -- drug effects
- Cell Survival -- drug effects
- Depsipeptides
- Diamines -- pharmacokinetics
- Drug Interactions
- Guanosine Triphosphate -- metabolism
- Mice
- Mitotic Index -- drug effects
- Molecular Sequence Data
- Oligopeptides -- pharmacology
- Organophosphorus Compounds -- pharmacokinetics
- Thiazoles -- pharmacology
- Tubulin -- metabolism
- Tumor Cells, Cultured -- drug effects
- Vinca Alkaloids -- metabolism
- Vincristine -- metabolism
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Publication Type: Comparative Study; Journal Article
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