In vitro and in vivo characterisation of Lu AF64280, a novel, brain penetrant phosphodiesterase (PDE) 2A inhibitor: potential relevance to cognitive deficits in schizophrenia. [electronic resource]
Producer: 20150804Description: 3151-67 p. digitalISSN:- 1432-2072
- Animals
- Antipsychotic Agents -- pharmacokinetics
- Avoidance Learning -- drug effects
- Behavior, Animal -- drug effects
- Cognition Disorders -- etiology
- Cyclic GMP -- metabolism
- Cyclic Nucleotide Phosphodiesterases, Type 2 -- antagonists & inhibitors
- Excitatory Amino Acid Antagonists -- pharmacology
- Heterocyclic Compounds, 4 or More Rings -- pharmacokinetics
- Hippocampus -- metabolism
- Humans
- Hyperkinesis -- chemically induced
- Male
- Mice
- Mice, Inbred DBA
- Phencyclidine -- antagonists & inhibitors
- Phosphodiesterase Inhibitors -- pharmacokinetics
- Rats
- Recognition, Psychology -- drug effects
- Recombinant Proteins
- Schizophrenia -- complications
- Schizophrenic Psychology
- Sensory Gating -- drug effects
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Publication Type: Journal Article
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