bba, a synthetic derivative of 23-hydroxybutulinic acid, reverses multidrug resistance by inhibiting the efflux activity of MRP7 (ABCC10). [electronic resource]
Producer: 20140508Description: e74573 p. digitalISSN:- 1932-6203
- ATP Binding Cassette Transporter, Subfamily B
- ATP Binding Cassette Transporter, Subfamily B, Member 1 -- genetics
- Adenosine Triphosphate -- metabolism
- Antineoplastic Agents -- metabolism
- Cell Line, Tumor
- Drug Resistance, Multiple -- genetics
- Drug Resistance, Neoplasm
- Gene Expression
- HEK293 Cells
- Humans
- Inhibitory Concentration 50
- Multidrug Resistance-Associated Proteins -- antagonists & inhibitors
- Paclitaxel -- metabolism
- Pentacyclic Triterpenes
- Protein Transport -- drug effects
- Triterpenes -- chemistry
- Betulinic Acid
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Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
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