CTA095, a novel Etk and Src dual inhibitor, induces apoptosis in prostate cancer cells and overcomes resistance to Src inhibitors. [electronic resource]
Producer: 20140923Description: e70910 p. digitalISSN:- 1932-6203
- Adenosine Triphosphate -- metabolism
- Animals
- Apoptosis -- drug effects
- Benzofurans -- pharmacology
- Binding Sites
- Cell Movement -- drug effects
- Cell Proliferation -- drug effects
- Disease Models, Animal
- Drug Resistance, Neoplasm -- genetics
- Enzyme Activation -- drug effects
- Human Umbilical Vein Endothelial Cells -- drug effects
- Humans
- Male
- Mice
- Models, Molecular
- Phosphorylation -- drug effects
- Prostatic Neoplasms -- metabolism
- Protein Binding
- Protein Conformation
- Protein-Tyrosine Kinases -- antagonists & inhibitors
- Proto-Oncogene Proteins c-akt -- metabolism
- Proto-Oncogene Proteins c-bcl-2 -- antagonists & inhibitors
- Proto-Oncogene Proteins c-myc -- antagonists & inhibitors
- Quinoxalines -- pharmacology
- STAT3 Transcription Factor -- metabolism
- Signal Transduction -- drug effects
- Xenograft Model Antitumor Assays
- src-Family Kinases -- antagonists & inhibitors
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Publication Type: Journal Article; Research Support, N.I.H., Extramural
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